プロフィール詳細

プロジェクトを作成

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Dr. Harish K.に依頼

India

Drug Discovery Medicinal Chemist with more than 10 years experience in Pharmaceutical Industry and Academia

プロフィール概要

Pharmaceutical Medicinal Chemist, Drug Discovery, Drug Design, Computer Aided Drug Design

専門分野

• ☆ Chemoinformatics
• ☆ Green Chemistry
• ☆ Computational Chemistry
• ☆ Biochemistry
• ☆ Antioxidants
• ☆ Pharmacy
• ☆ Pharmacy Education
• ☆ Clinical Pharmacy
• ☆ Drug Discovery
• ☆ High Throughput Screening (HTS)
• ☆ Drug Target Identification
• ☆ Hit-to-Lead & Lead Optimization
• ☆ Phenotypic Assays
• ☆ High Content Screening/Imaging
• ☆ Medicinal Chemistry
• ☆ Drug Design
• ☆ Combinatorial Chemistry
• ☆ Structure-Activity Relationship (SAR) Studies
• ☆ Drug Development
• ☆ Drug Formulation
• ☆ Small Molecule Drug Development
• ☆ Drug Substance Characterization
• ☆ Bioanalytical Testing
• ☆ Drug Stability Testing
• ☆ Preclinical ADME/PK/PD
• ☆ Drug-Drug Interactions
• ☆ Preclinical Research
• ☆ Preclinical Pharmacology
• ☆ Drug Efficacy Testing
• ☆ In vitro Diagnostics
• ☆ In vitro Diagnostic Design
• ☆ Medical Education
• ☆ Continuing Medical Education (CME)
• ☆ Health Informatics
• ☆ Positron Emission Tomography (PET)
• ☆ Complementary & Alternative Medicine
• ☆ Herbal Medicine
• ☆ Traditional Medicine
• ☆ Ayurveda
• ☆ Drug Delivery Technologies
• ☆ Pharmaceutical Technology

サービス

• Writing
• Research
• Consulting
• Product Development

Writing Technical Writing, Creative Writing, Newswriting, General Proofreading & Editing, Translation

Research Market Research, User Research, Meta-Research, Feasibility Study, Technology Scouting, Fact Checking, Gap Analysis, Scientific and Technical Research

Consulting Business Strategy Consulting, Scientific and Technical Consulting

Product Development Formulation, Stability/Shelf Life Testing

職務経験

HOD and Associate Professor

DY Patil Deemed to be University School of Pharmacy

1月 2022 - 現在

Associate Professor and Researcher

School of Pharmacy, D Y Patil Deemed to be University, Navi Mumbai, India

1月 2022 - 現在

Assistant Professor

Oriental College of Pharmacy

12月 2020 - 1月 2022

Assistant Professor

Shobhaben Pratapbhai Patel School of Pharmacy & Technology Management, SVKM's NMIMS University

4月 2017 - 7月 2020

Assistant Professor

C. U. Shah College of Pharmacy, SNDT University

6月 2016 - 12月 2016

Lecturer

Gahlot Institute of Pharmacy, Mumbai University

10月 2008 - 4月 2011

学歴

Ph.D.(Tech.)

Institute of Chemical Technology - India

4月 2011 - 12月 2017

認定資格

• Registered Pharmacist

  Pharmacy council of India

  10月 2006 - 現在

出版物

JOURNAL ARTICLE

(2020). Studies on spectral characterization and solubility of hydroxypropyl β-cyclodextrin/iloperidone binary and ternary complexes using different auxiliary agents . Journal of Molecular Structure.

(2019). Molecular dynamic simulations on an inhibitor of anti-apoptotic Bcl-2 proteins for insights into its interaction mechanism for anti-cancer activity . Journal of Biomolecular Structure and Dynamics.

(2019). Tetrahydrocurcumin-loaded vaginal nanomicrobicide for prophylaxis of HIV/AIDS: in silico study, formulation development, and in vitro evaluation . Drug Delivery and Translational Research.

(2019). Evaluation of phytopolyphenols for their gp120-CD4 binding inhibitory properties by in silico molecular modelling & in vitro cell line studies . Current HIV Research.

Kundaikar, Harish, Khambete, Mihir, Raju, Archana, Lonkar, Sachin, Degani, Mariam, Ray, Mukti Kanta (2019). Design and synthesis of 5-(5-nitrothiophen-2-yl)-3-phenyl-4,5-dihydro-1H-pyrazole derivatives with improved solubility and potential antituberculosis activity . Chemical Biology & Drug Design.

Anantram, A., Janve, M., Degani, M., Singhal, R., Kundaikar, H.(2018). Homology modelling of human divalent metal transporter (DMT): Molecular docking and dynamic simulations for duodenal iron transport . Journal of Molecular Graphics and Modelling. 85. Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 145-152.

Khambete, M., Kundaikar, H., Raju, A., Lonkar, S., Degani, M., Ray, M.K.(2018). Design and synthesis of 5-(5-nitrothiophen-2-yl)-3-phenyl-4,5-dihydro-1H-pyrazole derivatives with improved solubility and potential antituberculosis activity . Chemical Biology and Drug Design.

Kundaikar, Harish, Anantram, Aarti, Janve, Madhura, Degani, Mariam, Singhal, Rekha (2018). Homology modelling of human divalent metal transporter (DMT): Molecular docking and dynamic simulations for duodenal iron transport . Journal of Molecular Graphics and Modelling.

Bulani, V.D., Kothavade, P.S., Kundaikar, H.S., Gawali, N.B., Chowdhury, A.A., Degani, M.S., Juvekar, A.R.(2016). Inclusion complex of ellagic acid with β-cyclodextrin: Characterization and in vitro anti-inflammatory evaluation . Journal of Molecular Structure. 1105. Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 308-315.

Bulani, Vipin D., Kothavade, Pankaj S., Kundaikar, Harish S., Gawali, Nitin B., Chowdhury, Amrita A., Degani, Mariam S., Juvekar, Archana R. (2016). Inclusion complex of ellagic acid with beta-cyclodextrin: Characterization and in vitro anti-inflammatory evaluation . Journal of Molecular Structure.

Bulani, Vipin D., Kothavade, Pankaj S., Nagmoti, Dnyaneshwar M., Kundaikar, Harish S., Degani, Mariam S., Juvekar, Archana R. (2015). Characterisation and anti-inflammatory evaluation of the inclusion complex of ellagic acid with hydroxypropyl-beta-cyclodextrin . Journal of Inclusion Phenomena and Macrocyclic Chemistry.

Kundaikar, H.S., Sancheti, J.S., Jain, P.D., Degani, M.S., Sathaye, S.(2015). Docking studies and pharmacological evaluation of antiepileptic activity of phytoconstituents . Medicinal Chemistry Research. 24. (8). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 3296-3304.

Gangurde, A.B., Kundaikar, H.S., Javeer, S.D., Jaiswar, D.R., Degani, M.S., Amin, P.D.(2015). Enhanced solubility and dissolution of curcumin by a hydrophilic polymer solid dispersion and its insilico molecular modeling studies . Journal of Drug Delivery Science and Technology. 29. Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 226-237.

Bulani, V.D., Kothavade, P.S., Nagmoti, D.M., Kundaikar, H.S., Degani, M.S., Juvekar, A.R.(2015). Characterisation and anti-inflammatory evaluation of the inclusion complex of ellagic acid with hydroxypropyl-β-cyclodextrin . Journal of Inclusion Phenomena and Macrocyclic Chemistry. 82. (3). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 361-372.

Avinash B. Gangurde, Harish S. Kundaikar, Sharadchandra D. Javeer, Divakar R. Jaiswar, Mariam S. Degani, Purnima D. Amin (2015). Enhanced solubility and dissolution of curcumin by a hydrophilic polymer solid dispersion and its insilico molecular modeling studies . Journal of Drug Delivery Science and Technology.

Kundaikar HS, Degani MS (2015). Insights into the Interaction Mechanism of Ligands with A42 Based on Molecular Dynamics Simulations and Mechanics: Implications of Role of Common Binding Site in Drug Design for Alzheimer's Disease . Chemical Biology & Drug Design.

Kundaikar, H.S., Degani, M.S.(2015). Insights into the Interaction Mechanism of Ligands with Aβ42 Based on Molecular Dynamics Simulations and Mechanics: Implications of Role of Common Binding Site in Drug Design for Alzheimer's Disease . Chemical Biology and Drug Design. 86. (4). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 805-812.

Kundaikar, H.S., Agre, N.P., Degani, M.S.(2014). Pharmacophore based 3DQSAR of phenothiazines as specific human butyrylcholinesterase inhibitors for treatment of Alzheimer’s disease . Current Computer-Aided Drug Design. 10. (4). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 335-348.

Kundaikar, Harish S., Agre, Neha P., Degani, Mariam S. (2014). Pharmacophore Based 3DQSAR of Phenothiazines as Specific Human Butyrylcholinesterase Inhibitors for Treatment of Alzheimer's Disease . Current Computer-Aided Drug Design.

Kundaikar, H.S., Agre, N.P., Degani, M.S.(2014). Pharmacophore based 3DQSAR of phenothiazines as specific human butyrylcholinesterase inhibitors for treatment of Alzheimer’s disease . Current Computer-Aided Drug Design. 10. (4). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 335-348.

Vikas N. Telvekar, Kavit N. Patel, Harish S. Kundaikar, Hemchandra K. Chaudhari (2008). A novel system for the synthesis of nitriles from aldehydes using aqueous ammonia and sodium dichloroiodate . Tetrahedron Letters.

Telvekar, V.N., Kundaikar, H.S.(2008). GPR40 Carboxylic Acid Receptor Family and Diabetes: A New Drug Target . Current Drug Targets. 9. (10). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 899-910.

Telvekar, V.N., Patel, K.N., Kundaikar, H.S., Chaudhari, H.K.(2008). A novel system for the synthesis of nitriles from aldehydes using aqueous ammonia and sodium dichloroiodate . Tetrahedron Letters. 49. (14). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 2213-2215.

V. Telvekar, H. Kundaikar (2008). GPR40 carboxylic acid receptor family and diabetes: a new drug target . Current Drug Targets.

Telvekar, V.N., Kundaikar, H.S., Patel, K.N., Chaudhari, H.K.(2008). 3-D QSAR and molecular docking studies on aryl benzofuran-2-yl ketoxime derivatives as candida albicans N-myristoyl transferase inhibitors . QSAR and Combinatorial Science. 27. (10). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1193-1203.

Vikas N. Telvekar, Harish S. Kundaikar, Kavit N. Patel, Hemchandra K. Chaudhari (2008). 3-D QSAR and Molecular Docking Studies on Aryl Benzofuran-2-yl Ketoxime Derivatives as <i>Candida albicans</i> N-myristoyl transferase Inhibitors . QSAR & Combinatorial Science.