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プロフィール詳細
Dr. Kalpana T.に依頼
India
PhD in Pharmaceutical Chemistry experienced in writing and publishing 21 scientific articles in reputed journals.
プロフィール概要
専門分野
サービス
職務経験
Assistant Professor
Bharati Vidyapeeth's College of Pharmacy
1月 2021 - 現在 ![]()
PhD student & Research Fellow
Bharati Vidyapeeth's College of Pharmacy
9月 2017 - 1月 2021 ![]()
学歴
PhD
Bharati Vidyapeeth's College of Pharmacy, Navi Mumbai, India
1月 2017 - 1月 2021
認定資格
- 認定資格の詳細は未入力です。
出版物
JOURNAL ARTICLE
Kalpana Tilekar, Markus Schweipert, Niklas Jänsch, Neha Upadhyay, Ewelina Wozny, Sidra Basheer, Eva Wurster, Marlene Müller, Ramaa C S, Franz-Josef Meyer-Almes(2021). Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4 . Pharmaceuticals. 14. (10). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1032. {MDPI} {AG}
Kalpana Tilekar, Markus Schweipert, Niklas Jänsch, Neha Upadhyay, Ewelina Wozny, Sidra Basheer, Eva Wurster, Marlene Müller, Ramaa C S, Franz-Josef Meyer-Almes (2021). Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4 . Pharmaceuticals.
Upadhyay, N., Tilekar, K., Loiodice, F., Anisimova, N.Y., Spirina, T.S., Sokolova, D.V., Smirnova, G.B., Choe, J.-Y., Meyer-Almes, F.-J., Pokrovsky, V.S., et al.(2021). Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy . Bioorganic Chemistry. 107.
Kalpana Tilekar, Neha Upadhyay, Jessica D. Hess, Lucasantiago Henze Macias, Piotr Mrowka, Renato J. Aguilera, Franz-Josef Meyer-Almes, Cristina V. Iancu, Jun-yong Choe, C.S. Ramaa(2020). Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential . European Journal of Medicinal Chemistry. 202. Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 112603. Elsevier {BV}
Tilekar, K., Upadhyay, N., Meyer-Almes, F.-J., Loiodice, F., Anisimova, N.Y., Spirina, T.S., Sokolova, D.V., Smirnova, G.B., Choe, J.-Y., Pokrovsky, V.S., et al.(2020). Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents . ChemMedChem. 15. (19). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1813-1825.
Tilekar, K., Upadhyay, N., Hess, J.D., Macias, L.H., Mrowka, P., Aguilera, R.J., Meyer-Almes, F.-J., Iancu, C.V., Choe, J.-Y., Ramaa, C.S.(2020). Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential . European Journal of Medicinal Chemistry. 202.
Tilekar, K., Upadhyay, N., Jänsch, N., Schweipert, M., Mrowka, P., Meyer-Almes, F.J., Ramaa, C.S.(2020). Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines . Bioorganic Chemistry. 95.
Joshi, H., Patil, V., Tilekar, K., Upadhyay, N., Gota, V., Ramaa, C.S.(2020). Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib . Bioorganic and Medicinal Chemistry Letters. 30. (23).
Upadhyay, N., Tilekar, K., Jänsch, N., Schweipert, M., Hess, J.D., Henze Macias, L., Mrowka, P., Aguilera, R.J., Choe, J.-Y., Meyer-Almes, F.-J., et al.(2020). Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation . Bioorganic Chemistry. 100.
Tilekar, K., Upadhyay, N., Schweipert, M., Hess, J.D., Macias, L.H., Mrowka, P., Meyer-Almes, F.-J., Aguilera, R.J., Iancu, C.V., Choe, J.-Y., et al.(2020). Permuted 2,4-thiazolidinedione (TZD) analogs as GLUT inhibitors and their in-vitro evaluation in leukemic cells . European Journal of Pharmaceutical Sciences. 154.
Tilekar, K., Upadhyay, N., Iancu, C.V., Pokrovsky, V., Choe, J.-Y., Ramaa, C.S.(2020). Power of two: combination of therapeutic approaches involving glucose transporter (GLUT) inhibitors to combat cancer . Biochimica et Biophysica Acta - Reviews on Cancer. 1874. (2).
Vora, D., Upadhyay, N., Tilekar, K., Jain, V., Ramaa, C.S.(2019). Development of 1,2,4-triazole-5-thione derivatives as potential inhibitors of enoyl acyl carrier protein reductase (Inha) in tuberculosis . Iranian Journal of Pharmaceutical Research. 18. (4). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1742-1758.
Kabir, A., Tilekar, K., Upadhyay, N., Ramaa, C.S.(2018). Novel anthraquinone derivatives as dual inhibitors of topoisomeras e 2 and casein kinase 2: In silico studies, synthesis and biological evaluation on leukemic cell lines . Anti-Cancer Agents in Medicinal Chemistry. 18. (11). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1551-1562.
Patil, V., Tilekar, K., Mehendale-Munj, S., Mohan, R., Ramaa, C.S.(2010). Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2,4- thiazolidinedione derivatives . European Journal of Medicinal Chemistry. 45. (10). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 4539-4544.
Ramaa, C.S., Tilekar, K.N., Patil, V.M.(2010). Liver cancer: Different approaches for targeting . International Journal of PharmTech Research. 2. (1). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 834-842.