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プロフィール詳細
プロジェクトを作成
★★★★★
☆☆☆☆☆
Dr. Kalpana T.に依頼
India

PhD in Pharmaceutical Chemistry experienced in writing and publishing 21 scientific articles in reputed journals.

プロフィール概要
専門分野
サービス
Writing Technical Writing
Research Market Research, User Research, Meta-Research, Feasibility Study, Gap Analysis, Gray Literature Search, Systematic Literature Review, Secondary Data Collection
Data & AI Statistical Analysis
職務経験

Assistant Professor

Bharati Vidyapeeth's College of Pharmacy

1月 2021 - 現在

PhD student & Research Fellow

Bharati Vidyapeeth's College of Pharmacy

9月 2017 - 1月 2021

学歴

PhD

Bharati Vidyapeeth's College of Pharmacy, Navi Mumbai, India

1月 2017 - 1月 2021

認定資格
  • 認定資格の詳細は未入力です。
出版物
JOURNAL ARTICLE
Kalpana Tilekar, Markus Schweipert, Niklas Jänsch, Neha Upadhyay, Ewelina Wozny, Sidra Basheer, Eva Wurster, Marlene Müller, Ramaa C S, Franz-Josef Meyer-Almes(2021). Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4 . Pharmaceuticals. 14. (10). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1032. {MDPI} {AG}
Kalpana Tilekar, Markus Schweipert, Niklas Jänsch, Neha Upadhyay, Ewelina Wozny, Sidra Basheer, Eva Wurster, Marlene Müller, Ramaa C S, Franz-Josef Meyer-Almes (2021). Mechanistic Insights into Binding of Ligands with Thiazolidinedione Warhead to Human Histone Deacetylase 4 . Pharmaceuticals.
Upadhyay, N., Tilekar, K., Loiodice, F., Anisimova, N.Y., Spirina, T.S., Sokolova, D.V., Smirnova, G.B., Choe, J.-Y., Meyer-Almes, F.-J., Pokrovsky, V.S., et al.(2021). Pharmacophore hybridization approach to discover novel pyrazoline-based hydantoin analogs with anti-tumor efficacy . Bioorganic Chemistry. 107.
Kalpana Tilekar, Neha Upadhyay, Jessica D. Hess, Lucasantiago Henze Macias, Piotr Mrowka, Renato J. Aguilera, Franz-Josef Meyer-Almes, Cristina V. Iancu, Jun-yong Choe, C.S. Ramaa(2020). Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential . European Journal of Medicinal Chemistry. 202. Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 112603. Elsevier {BV}
Tilekar, K., Upadhyay, N., Meyer-Almes, F.-J., Loiodice, F., Anisimova, N.Y., Spirina, T.S., Sokolova, D.V., Smirnova, G.B., Choe, J.-Y., Pokrovsky, V.S., et al.(2020). Synthesis and Biological Evaluation of Pyrazoline and Pyrrolidine-2,5-dione Hybrids as Potential Antitumor Agents . ChemMedChem. 15. (19). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1813-1825.
Tilekar, K., Upadhyay, N., Hess, J.D., Macias, L.H., Mrowka, P., Aguilera, R.J., Meyer-Almes, F.-J., Iancu, C.V., Choe, J.-Y., Ramaa, C.S.(2020). Structure guided design and synthesis of furyl thiazolidinedione derivatives as inhibitors of GLUT 1 and GLUT 4, and evaluation of their anti-leukemic potential . European Journal of Medicinal Chemistry. 202.
Tilekar, K., Upadhyay, N., Jänsch, N., Schweipert, M., Mrowka, P., Meyer-Almes, F.J., Ramaa, C.S.(2020). Discovery of 5-naphthylidene-2,4-thiazolidinedione derivatives as selective HDAC8 inhibitors and evaluation of their cytotoxic effects in leukemic cell lines . Bioorganic Chemistry. 95.
Joshi, H., Patil, V., Tilekar, K., Upadhyay, N., Gota, V., Ramaa, C.S.(2020). Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib . Bioorganic and Medicinal Chemistry Letters. 30. (23).
Upadhyay, N., Tilekar, K., Jänsch, N., Schweipert, M., Hess, J.D., Henze Macias, L., Mrowka, P., Aguilera, R.J., Choe, J.-Y., Meyer-Almes, F.-J., et al.(2020). Discovery of novel N-substituted thiazolidinediones (TZDs) as HDAC8 inhibitors: in-silico studies, synthesis, and biological evaluation . Bioorganic Chemistry. 100.
Tilekar, K., Upadhyay, N., Schweipert, M., Hess, J.D., Macias, L.H., Mrowka, P., Meyer-Almes, F.-J., Aguilera, R.J., Iancu, C.V., Choe, J.-Y., et al.(2020). Permuted 2,4-thiazolidinedione (TZD) analogs as GLUT inhibitors and their in-vitro evaluation in leukemic cells . European Journal of Pharmaceutical Sciences. 154.
Tilekar, K., Upadhyay, N., Iancu, C.V., Pokrovsky, V., Choe, J.-Y., Ramaa, C.S.(2020). Power of two: combination of therapeutic approaches involving glucose transporter (GLUT) inhibitors to combat cancer . Biochimica et Biophysica Acta - Reviews on Cancer. 1874. (2).
Vora, D., Upadhyay, N., Tilekar, K., Jain, V., Ramaa, C.S.(2019). Development of 1,2,4-triazole-5-thione derivatives as potential inhibitors of enoyl acyl carrier protein reductase (Inha) in tuberculosis . Iranian Journal of Pharmaceutical Research. 18. (4). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1742-1758.
Kabir, A., Tilekar, K., Upadhyay, N., Ramaa, C.S.(2018). Novel anthraquinone derivatives as dual inhibitors of topoisomeras e 2 and casein kinase 2: In silico studies, synthesis and biological evaluation on leukemic cell lines . Anti-Cancer Agents in Medicinal Chemistry. 18. (11). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 1551-1562.
Patil, V., Tilekar, K., Mehendale-Munj, S., Mohan, R., Ramaa, C.S.(2010). Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2,4- thiazolidinedione derivatives . European Journal of Medicinal Chemistry. 45. (10). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 4539-4544.
Ramaa, C.S., Tilekar, K.N., Patil, V.M.(2010). Liver cancer: Different approaches for targeting . International Journal of PharmTech Research. 2. (1). Microsoft.AspNetCore.Mvc.Localization.LocalizedHtmlString 834-842.